Free Letter - District Court of Delaware - Delaware


File Size: 117.6 kB
Pages: 4
Date: July 6, 2005
File Format: PDF
State: Delaware
Category: District Court of Delaware
Author: unknown
Word Count: 1,247 Words, 11,312 Characters
Page Size: 612 x 794 pts
URL

https://www.findforms.com/pdf_files/ded/7523/58-2.pdf

Download Letter - District Court of Delaware ( 117.6 kB)


Preview Letter - District Court of Delaware
Case 1:04—cv—00171-GI\/IS Document 58-2 Filed 07/06/2005 Page1 0f4

Case 1 :04—cv—00171-GI\/IS Document 58-2 Filed 07/06/2005 Page 2 0f 4
Ulliiitd States Paféllf ns; {11] Patent Number: 5,668,249
Long [45} Date of Patent: Nm. 26, 1991
[54} AQUEOUS RANZIIDHWE CONIPGSITIONS {56] ima-nm Cited
Sm*mzE¤ WH Em*“°*· Fon-zum: rxram nocxmzrws ‘
hI¥'£·'¢u£!¥2 R. m 15*772-; 11/1gs* Fung: _ l
{73] Assiwnc: gniesafjmay Ijnitsé, Landon, Ki¤¤6¤¤
{21} Appl. Nm mm Mn 0THE:~:f;:;1aL?é;sTIONS
. (sv;-sz .
Eu] Fiki M"` R, 1999 Chem. Abt. ·[l04}~E¤225€}Z (1986). ·
MMM U5- -'~r¤¥i¤¤¤• ¤·¤ mma mmksmmx 2. wwwa ·
{63] cmmum ¤r su. ug. wm Ap-. zu. am, mu- A=¤f¤==¤¤ £·wmiw—·g¤i¤¤¤ G¤¤¤=r
%•:§.;w§g u · Mmmm at se:. Ne E31.M1. Aww- »·¢¢¢¤¤ ¤#F¤¤¤·-B•¤¤¤ 1 ’i`!=¤¤¤¤ 1
’ ‘ sv; Amman
BQ] Fwd, Ananda hjmunm Ffh: subilityofnquacan fnrmulszicwufnnitidiuccwa
Doc. S2, 19Bé {GE] United E|\f£E ............... M 297II Inxpbhgn. an mawfh cuhlagcd by
[sz; zu. c¤.= ............"..... ........ ”.,.......“ mx was ¤¤= ·¢¤if•¤¤ ¤f=¤=¤¤1·
[::2} U.S. CL .................................................... 514/{TI
{58} Field nf Search ..q.........,.................... 514/661. HI $3 China, No Dnwlmt

Case 1:04—cv—00171-GI\/IS Document 58-2 Filed 07/06/2005 Page 3 0f 4
1 5,063,249 ` 2
Aprefurcd ¤¤h¤dim¤ntafth¢i¤v¤as5¢misx¤uq¤s—
AQUEOUS RAHIHDINE COMPQSIHONS umfcrmuhzbnfnrmdmmmmrmm. smhgfm-muh-
S}`AB!I.!Z'EDV\’IT§iE!1IAIWOL ticnmsyccmyriscraniddimndfurmcwmndim
physkzlugiuiiy anczpuhk axudiuchmdin u.·•m·.¢th·
ncmtimmiuu axfapplicuiou Ser. 5 mn}. n preservative and t viscosity enhancing agent.
Nc. 07,/344.620. 514% Ap:. 25, 1985, now nbmdcnzd, Prdmbiy the required pH of the fnnnumicn is ¤h-
whlch is a ccutimudmi ¤{S¤. Nm. 07JI3l,4·$2, fixed :·i§¤dbytb¤¤:c¤hppdr·¤:ristcb1•i¥¢§1\;af1!s.Qpti¤¤s¥!y
Dec. II, 19|7, now abandoned. cumpnsiticn may nnmain u ccmvnmi
Thzprucnt invasion mhteiw n pisumxzvtical I0 ¢xcipi¢¤¤u•chuaswe¤te¤e:r.n¤sv¤¤:and!c:¤•-
mv { _ °E¤M¤ph¤ of miubl: pxnavulvu iactudn un cr
[N-[2·[{[5~(dim:thyh¤i¤o)m¤hyi-2- more alkyl lzydrmybcnxmu such as mcxhyi, efhyi.
fur¤yf]mc¢I1yI]d1i¤]¤3¤yI]·N'·;e:hyL2·1i¤¤-:;§>3c,·$ pmpyl and/cgfbutyi hydryxybgzmnm. * u.
d¤4:xR:¤da:¢§i£ak¥y¤;um N:*$ch:d¢X¤thmg¤m.s¤:ti=¤¤E;ty¤cr¤Lsa¤r§¤r»
1565966.In mimspecimazionxbcreisrzfezemnemiiquid ¤¤K¤l¤•¤r1¤·Ivnt£vn•¤¤hatc¤*b¤¤ym¤shy}c¤B¤1¤•c ur
fcrmulaeiomfurmsludpnnmuxlpdmiaismzknsgnd n·•!ttb¤x·¤¤l'ofnC;..••1k3·|and/¤rnh;·d:¤xy~C;.•all:y\
xbueisnducriptioucfmnquauubundfnrmulxtim ¢th¤’¤f¤¢Hui¤•¢$uch¤m¢tI¤y1¤¢1I¤I¤••,e:I:y1¤é1v-
fcrimruveacuuueanduuxhucfmmdaymphosh so %¤•¤. hydmxydhyicdlulca, hyd:-cxypmpyludiuluen,
ufnbac mrmumiunaccuainnésutticinunhyamcsasaria hy¤r¤¤ycr!:y mn hy¤.n¤xypr¤py$u»·
n¤idl¤•¤hiev¢apH¤i'5.0:¤dth::yr¤;¤n1so¢¤¤· !hy?¤d]¤l0••. _ _ _
¤i¤cd5¤1bimis¤1uti¤¤BPCa¤dn¤nmnu:¤qui;-¤d, B¤mpi¤_¤fsumbh¤w¤¤.¤x?¤s mdudznmhum
BritlIhP1¤¤¤£AppIica¤i¤¤ No.GB 2I42¤¤Ad;- I '
mn'hu.squa¤n»bnmdf¤a¤¤1n:i¤¤4 $-¤m;»Ia•¤£•u¤:bl•!hy¤mm5•qs¤¤;»¤1¤d¤*¤»s
dineaa-ad/¤1·¤¤:m-mnnctiuphydoiqgigauy weep;. ¤•v¤¤¤s¤¤ka•pppp¤1¤m:,{t{v¤uymg qua:.
•b1¤sai¤1b¤r¤¤fh.nvin;•pHu¢irhi¤th¤n§£‘§e6.5-7.$, d°';N ¤f¤m;d¤¢m:?swd§¤gmw`;:·
{nth: sp¤¤:.fi¤a¤¤¤' ' thu! zefexuua ` ` fom-mIa» ¤ M
r5¤¤»;¤r¤ra1•ndp•z:¤z:11 md¢b¤¤ ¤=¤I¢2°—*€¤¤xP¤l0¤L¥¤¢¤¤mv!¤1¤·1<¤m|v¤
amuamplucfaqumufcmuindcnafnrinwsvzuou m¤¥•¤¤¥*P*¤i¤¤¥¤’?Y*$°¤§i¤¤J0¤¤¥*$¤*¤·
¤¤t!¤¤l¤•c.T'h¤¢f¤rmuh5¤aa¤¤~¤uS¤¤¤i:kii¤;3° 'n\¢¤¤¤¤¤l¤i'¤thm¤!B1thcf¤r¤uIat§¤¤f¤rox;}
by;¤ch}¤rida¤d;r¢b¤f1'¤¤|m•p}i¤f;pp;q;$;¤gp3y ¤pn¤¤d}1np¤r¤m¤g¤ uhh; com-
1 me rm awww me rmmmm 9** f¤¤¤¤·i•¤i¤¤ ¤¤ ¤ wwvwfm wir. ir prefera-
»1·¤¤¤¤¤a»p1.¢¤¤1¤¤»¤¤a¤¤¤¤1¤;¤¤¤¤.1¤¤¤¤¤n;¤¤1¤· '=¥1*¢W¤¤·¤¤•¤¤=2-5¤¤1¤*1¤·•¤<¥¤=¤¤¤s~·¤i¤¤i¤r|:
i1¤•tii¤nthcf¤rmu1•d»¤¤ds¤¤¤¤uk;¤hy¤3;¤;)»p4·°py1. is ¤¤_¤;*:¤15¤E\';_6.]1n¤1g‘;sp¤¤$dlyT~I:b;;ti¤thcf
mtu:} · · enhandua tmbim _Vi¤¤l2 S Q1`-
a¤-vn§v¤(pu:“1z:)Tz manning agent m¤mi¤¤•wi11p¤·¢£¢nbi¥B¤s¤1H¤i:¤xn¤giv¤¤sc1¤ti¤¤
-· |.,“,,,,; ;gc,,,, ,, , withav§s¤¤¤it·yi¤the:•n;:¤fI0m1{Il¢¤uip¢mlu¤L
linuecouxpcmhzm an iv ar wmv . . .
Hf¤¤v¤·th¤•ei¤§z·id•hPa1¤¤tN0.!§45$966.
We have mw wpzidugly found thnithz nmmey gm °°m'f¤i¥¤uY?*`¤P¤¤db¥¤¤&8¤Q4¤¢¤N?0}¤!{0¤0f
¤¤inidh1¢i¤•qu¢·¤n¤ m;6¤?;¤;¢¤¤;;,¤. ¤¤f¤di¤¤a§“}d;m¤¤¤w‘¥;r¤dm pc§ui¥
uw aquacmstned tion cnhsimiuir- _ ‘“‘_ P
mmmymruwmymmmwagrmmmmd gjxwim nzmumuunumuupemmamvww
cthmul the utf ¤*h*¤d¤ *8***- .
*5 ThlIq¤¤¤¤f¤¤‘¤¤hti0qin¤:c¢;d§n-gt¤thgi¤v¤1i¤¤
qsmmdumwuakmmnummmumgnmu. ;¢:h¤¥=¥¤•¤¥v¤1~=1:;¤¤¤¤manm¤¤¤¤¤i¤¤=¤f¤=¤¤f
x ,,,'““,‘;§f' ,j',°§ °"§’,,,;,,¤“°7”",,;,,,,L` ’° $Tk¤3“11lx1¤== " °`,·,,,"Z in itiuanudva uampk ¤n r¤m¤ms¤¤ »¤¤¤¤sx¤; uz
mgm- P,.q,.,,d,_,·"·,,¥;¤ in of paw mh tbeinvnénahafnuuwglutbisusmpkzhcrdnéve
gsuirissziubtetuuummumgpszuemwm 3, s¤¤1¤¤¤i¤¢¤¤fn¤iddi¤chyd:¤¤h3¤ndeaa¤¢¤¢¤¤rr¢»
emxmmummmvmmpwmm ·~¤··=¤·¤¤¥¤·=¤¤=¤~=f<=·¤¤*·¤¤¤1=¤·v¥*¤¤f¤vv¤¤=*·
0 uwrucipamsmmcxuencqzaennannzmdmiaidim ¤’”·*YY~ 1
a¤£;rphy•i¤|cgi¤3}ym¤¤px¤b£¢ahn¤h¤¤¤&
smcuntcfnhauoiprcscntintlacfcrmulaécair
mchthuhfwddu Mmmdmmw 8 :»¤¤»¢¤u¤q¤us¤¢¤¤1»s¤»;1s¤¤y1¤¤n
s¤b{ii:y.Pr¤f¢nb1yu»e•m·¤•¤n¤£nh¤¤4i¤ab¤¤¤¤»- sun
m¤1asi¤¤.i¤withh1thc—r•¤g¤2.55¢¤I095.andm¤ze haunt
pu1ic¤1sr£y§sb¢¤vo¤31¤$0%wfv,m¤r¤¤spa¤ial1y W5
T--8% wv, w usc
Prcfmeu ccmpcrnsnu accmdiug ua the iuveminu :
aret.b¤•ei¤wh$¤hthepH0ftb¢aq¤v¤¤•fcru:uhrin¤£¤ s·¤¤¤aq••¤¤u qs
within the mp 6.5 za 7.5. pnnicuhriy $.8 rn 7.4 and Www nv
me ¤p¤¤s.¤y1m1.s.11¤¤mq¤»ar¤¤px¤¢m»r¤¢m¤·
hmiangryeofaaglliobuinedhythcunsofauiublcbutvn in
aiu cum pcami ···- dihydmgcu cnbcphm- Ichim:
pluumd discéium hydrogen cnhophosphatc ur citric 1. A phnrmuzulicd compqdtinm which innaquemu
hydmgm mhopbmphau. furmulnciun for mal uf an effective

Case 1:04—cv—00171-GI\/IS Document 58-2 Filed 07/06/2005 Page 4 0f 4
3 5,068,249 ‘
axmxmnfzmizidiue md/an-¤m¤:m¤r¤pbysin1¤;$· 8.Aphu-mmcuti¤s1comp¤sit$cnu:1nim¤dindnim
cuilyaucepnbtnanszhercoiaidfomunnsunmmprk- 1.wh¤¤i¤¤h:¤£fmiv¤nmmm¤k20-évumgxmiddinz
i¤gnmbiii:i¤g¢!!'¤c:iv¢u¤¤u¤tcfcd1anoi•uds•.id pcrwmlduaccxprzsacdaafrecbxsa
composition h•vi:¤g¢pHinthcn¤g¤¤f6.5·7J. thphnrmwcuxinlcnmpcsidanuchimcdiasdiha
2.Apiu:ma¤¤mi¤l¤¤mp¤¤iri¤¤¤¤¤¤:di:ag¢¤c3nim s 1,wh¤r¢i¤ahe¢H‘c¤iv¢am¤xmti»1¤—2DGmgrmitid1¤¢
1 containing 2.5% to 10% w:§gh1fv¤1nnm¤.¤ahm¤l pexiihnldnsezxpruscdufrccbne. _
buedcnthecompletsfcrmuiation. · 10.A ¤¤mp0•ir.icnascIai:¤c¢iin¤lai¤¤
$.Ap3za11mu¤¤ulI¤a! composition avccmiinghucinim 1,,wh¤¤&¤th:;R';c¢iv¤¤m¤u¤t§a1§0¤x;rnnis§di:¤•;:•r
I¢¤a¤u£1zi¤g7$et¤8‘$¥¤ weighzfvolume uhmciuued lihnlduscuprusudusfxeebasn.
cudaecumpietcfcmuiaxion. za 1I.A ¤¤mpui¢i¤nwhicbi:¢¤»q¤¤·
·t.A c¤mpcsiti¤»¤ amczdingtoclsim uufarmuladun nfnnitidincmziubic for nnlanhniuis-
1mwim;•pHi¤:h¤r¤¤g¤6.8m1.4. mt$¤¤¤:•¤¤i¤i¤sl50mgn¤&¤:tincv¤ri0m1d¤•¤ ‘
5.A ¤nmpné2.i¤nx¤:¤rdi¤gm¤$nim ¤pr¤•¤dufr¢cbs¢,¤.id£onnu1ati¤¤h•vb1g•pHi¤ _ .
11uvhzgapHinth¤:m5:7.01¤7.3. the:mg¤7.0w7.3mdaln¤¤¤uni:s1ing7*H»¤¤§%
6.A. ¤0mpoeidcna¤¤¤:di¤g¤¤ckim is w¢ig1:u‘v¤§¤mc¤1ha¤¤1b¤ed¤¤dac¤¤pi¤¤f¤w¤,¤l» `
1whe::i¤n%dpI—Iiwbui¤¤dby¢!»:1ue¤4butf¤u2¤. zion. _
‘7.Aph.um;¤eutical¤¤¤p¤¤i:i¤¤ac¤¤rdingt¤¤l¤kn Ilapbumaccutimicomposixinnaccordinsznciaim
Ipregarndusing rauiddincinthcfnrmnfthzhydrv uwh:mi¤nidpH§m3euin¢dbyth:1¤e0fb¤¤”¤a1u.
chkxidcsdt. " ‘ " ‘ ’
29
za
- J5 `
ac
as
_ _ S0
ss
60
ss

Case 1:04-cv-00171-GMS

Document 58-2

Filed 07/06/2005

Page 1 of 4

Case 1:04-cv-00171-GMS

Document 58-2

Filed 07/06/2005

Page 2 of 4

Case 1:04-cv-00171-GMS

Document 58-2

Filed 07/06/2005

Page 3 of 4

Case 1:04-cv-00171-GMS

Document 58-2

Filed 07/06/2005

Page 4 of 4